The project was financially supported by the National Natural Science Foundation of China (Grant Nos. 21476065, 21571060, 21725602) and the Fundamental Research Funds for the Central Universities (Hunan University). CTA thanks HNU for an adjunct professorship.
机构署名：
本校为通讯机构
院系归属：
医学院
中医学院
摘要：
AbstractCopper‐catalyzed cross‐dehydrogenative esterification of readily available N‐heteroaryl methanes with acids has been realized in good to excellent yields of target products. Through simple regulation of acid loading, it is possible to achieve mono‐ or di‐esterification of the methyl group with high chemoselectivity. The protocol is suitable for a wide scope of substrates and exhibits high step efficiency and atom economy. It is envisaged that this radical‐promoted one‐pot dual functionalization of C(sp3)−H bond is a general and ...
